CAS号:802539-81-7
品名:4,5-二氢-n,1,4,4-四甲基-8-[[4-(4-甲基-1-哌嗪)苯基]氨基]-1H-吡唑并[4,3-h]喹唑啉-3-羧酰胺N,1,4,4-tetramethyl-8-[4-(4-methylpiperazin-1-yl)anilino]-5H-pyrazolo[4,3-h]quinazoline-3-carboxamide
中文别名:4,5-二氢-n,1,4,4-四甲基-8-[[4-(4-甲基-1-哌嗪)苯基]氨基]-1H-吡唑并[4,3-h]喹唑啉-3-羧酰胺
英文别名:Milciclib[INN];N,1,4,4-tetramethyl-8-(4-(4-methylpiperazin-1-yl)phenylamino)-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide;Milciclib;
分子式:C25H32N8O
分子量:460.575
精确质量:460.27
Psa:94.7
MDL号:MFCD17169990
密度:1.33 g/cm3
简介:PHA-848125isacyclindependentkinase(CDK)inhibitor.OralPHA-848125showedantitumoractivityviadualtargetingofcyclin-dependentkinaseandtropomyosinreceptorkinasefamiliesinhumancarcinomacellandxenograftedmousemodelofcarcinoma.
细胞周期