CAS号:936091-14-4
品名:N-(1,1-二甲基乙基)-3-[[5-甲基-2-[[4-(4-甲基-1-哌嗪基)苯基]氨基]-4-嘧啶基]氨基]苯磺酰胺N-tert-butyl-3-[[5-methyl-2-[4-(4-methylpiperazin-1-yl)anilino]pyrimidin-4-yl]amino]benzenesulfonamide
中文别名:N-(1,1-二甲基乙基)-3-[[5-甲基-2-[[4-(4-甲基-1-哌嗪)苯基]氨基]-4-嘧啶]氨基]苯磺酰胺;
英文别名:N-(1,1-DIMETHYLETHYL)-3-[[5-METHYL-2-[[4-(4-METHYL-1-PIPERAZINYL)PHENYL]AMINO]-4-PYRIMIDINYL]AMINO]BENZENESULFONAMIDE;1M3;Kinome_702;N-tert-butyl-3-(5-methyl-2-(4-(4-methylpiperazin-1-yl)phenylamino)pyrimidin-4-ylamino)benzenesulfonamide;
分子式:C26H35N7O2S
分子量:509.667
精确质量:509.257
Psa:114.1
密度:1.25
沸点:703.1ºC at 760 mmHg
闪点:379ºC
简介:TG101209isaneffectivetyrosinekinaseinhibitoroftyrosinekinasesJAK2andJAK3(januskinase2/3),inducingcellarrestandapoptosisinleukemiacelllines.
JAK/STAT