内分泌与激素

CAS号：130663-39-7

品名：PD123319PD123319

中文别名：PD123319

英文别名：1-((4-(Dimethylamino)-3-methylphenyl)methyl)-5-(diphenylacetyl)-4,5,6,7-tetrahydro-1H-imidazo[4.5-c]pyridine-6-carboxyli;(6S)-1-[4-(Dimethylamino)-3-methylbenzyl]-5-(diphenylacetyl)-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridine-6-carboxylicacid;S-(+)-1-((4-(dimethylamino)-3-methylphenyl)methyl)-5-(diphenylacetyl)-4,5,6,7-tetrahydro-1H-imidazol(4,5-c)pyridine-6-carboxylicacid;pd123,319di(trifluoroacetate)salt;PD123,319;(3S)-9-[(4-DIMETHYLAMINO-3-METHYL-PHENYL)METHYL]-4-(2,2-DIPHENYLACETYL)-4,7,9-TRIAZABICYCLO[4.3.0]NONA-7,10-DIENE-3-CARBOXYLICACID;(S)-1-&<&<4-(dimethylamino)-3-methylphenyl&>methyl&>-5-(diphenylacetyl)-4,5,6,7-tetrahydro-1H-imidazo&<4,5-c&>pyridine-6-carboxylicacid;PD123,319DITRIFLUOROACETATE;

分子式：C31H32N4O3

分子量：508.611

精确质量：508.247

Psa：78.67

密度：1.22 g/cm3

沸点：775.8ºC at 760 mmHg

闪点：423ºC

储存条件：2-8ºC

蒸汽压：2.48E-25mmHg at 25°C

危险品标志：Xi

内分泌与激素

CAS号：851983-85-2

品名：Galeterone(3S,8R,9S,10R,13S,14S)-17-(benzimidazol-1-yl)-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15-decahydro-1H-cyclopenta[a]phenanthren-3-ol

中文别名：Galeterone

英文别名：(3S,8R,9S,10R,13S,14S)-17-(benzimidazol-1-yl)-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15-decahydro-1H-cyclopenta[a]phenanthren-3-ol

分子式：C26H32N2O

分子量：388.545

精确质量：388.251

Psa：38.05

UNII号：WA33E149SW

密度：

简介：Galeterone(TOK-001orVN/124-1)isanovelsteroidalantiandrogenunderdevelopmentbyTokaiPharmaceuticalsforthetreatmentofprostatecancer.Itpossessesauniquedualmechanismofaction,actingasbothanandrogenreceptorantagonistandaninhibitorofCYP17A1,anenzymerequiredforthebiosynthesisoftheandrogens.Itshowsselectivityfor17,20-lyaseover17-hydroxylase.