Enzastaurin Enzastaurin 1mg

CAS号：170364-57-5

品名：丁胺苯丙酮3-(1-Methyl-1H-indol-3-yl)-4-(1-(1-(pyridin-2-ylmethyl)piperidin-4-yl)-1H-indol-3-yl)-1H-pyrrole-2,5-dione

中文别名：恩扎妥林;2-氧杂-6-氮杂螺[3,3]庚烷草酸盐;3-(1-甲基-1H-吲哚-3-基)-4-(1-(1-(2-吡啶甲基)-4-哌啶基)-1H-吲哚-3-基)-1H-吡咯-2,5-二酮;

英文别名：3-(1-methylindol-3-yl)-4-[1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]indol-3-yl]pyrrole-2,5-dione;Enzastaurin;

分子式：C32H29N5O2

分子量：515.605

精确质量：515.232

Psa：72.16

MDL号：MFCD11040980

密度：1.34g/cm3

沸点：767.2ºC at 760mmHg

闪点：417.8ºC

折射率：1.722

蒸汽压：1.87E-23mmHg at 25°C

海关编码：2933990090

信号词：Warning

危险标志：GHS07

危险性描述：H302; H413

简介：Enzastaurinisasyntheticbisindolylmaleimidewithpotentialantineoplasticactivity.BindingtotheATP-bindingsite,enzastaurinselectivelyinhibitsproteinkinaseCbeta,anenzymeinvolvedintheinductionofvascularendothelialgrowthfactor(VEGF)-stimulatedneo-angiogenesis.Thisagentmaydecreasetumorbloodsupply,preventinggrowth.

用途：丝氨酸/羟丁氨酸激酋每抑制剂