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CAS:546-06-5
546-06-5
CAS号：546-06-5
品名：止泻木碱conessine
中文别名：地麻素;
英文别名：CONESSIN;Con-5-enin-3-amine,N,N-dimethyl-,(3β)-;WRIGHTINE;ROQUESSINE;NERVINE;NERIINE;ROGUESSINE;Conessine,N,N-Dimethyl-con-5-enin-3-amine;5-CONENIN-3BETA-DIMETHYLAMINE;1-Deazaadenosine;
分子式：C24H40N2
分子量：356.588
精确质量：356.319
Psa：6.48
UNII号：EZ38J9BBDF
密度：1.05g/cm3
沸点：450.4ºC at 760 mmHg
熔点：126-127ºC
闪点：199.6ºC
折射率：1.564
储存条件：Store at RT
简介：ConessineisasteroidalkaloidfoundinanumberofplantspeciesfromtheApocynaceaefamily,includingHolarrhenafloribunda,HolarrhenaantidysentericaandFuntumiaelastica.Itactsasahistamineantagonist,selectivefortheH3subtype(withanaffinityofpKi=8.27;Ki=~5nM).ItwasalsofoundtohavelongCNSclearancetimes,highblood-brainbarrierpenetrationandhighaffinityfortheadrenergicreceptors.
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