CAS号:700874-72-2
品名:LY2157299;4-[5,6-二氢-2-(6-甲基-2-吡啶基)-4H-吡咯并[1,2-b]吡唑-3-基]-6-喹啉甲酰胺2-(6-methylpyridin-2-yl)-3-(6-aminocarbonylquinolin-4-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole
中文别名:LY2157299;4-[5,6-二氢-2-(6-甲基-2-吡啶基)-4H-吡咯并[1,2-b]吡唑-3-基]-6-喹啉甲酰胺
英文别名:6-[2-(6-Methylpyridin-2-yl)-acetyl]quinoxaline;2-(6-methyl-pyridin-2-yl)-3-(6-amido-quinolin-4-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole;2-(6-Methyl-pyridin-2-yl)-1-quinoxalin-6-yl-ethanone;
分子式:C22H19N5O
分子量:369.419
精确质量:369.159
Psa:86.69
MDL号:MFCD12923319
密度:1.409 g/cm3
沸点:619.004ºC at 760 mmHg
闪点:328.162ºC
简介:LY2157299isaTGF-βtypeIreceptorkinaseinhibitor.LY2157299hasbeenusedtoinhancechemotherapyactionagainsttriplenegativebreastcancer(TNBC).
TGF-beta/Smad