CAS:1346574-57-9
1346574-57-9
CAS号：1346574-57-9
品名：GSK1261-[(2S)-butan-2-yl]-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-methyl-6-(6-piperazin-1-ylpyridin-3-yl)indole-4-carboxamide
中文别名：GSK126
英文别名：(S)-1-sec-butyl-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-3-methyl-6-(6-(piperazin-1-yl)pyridin-3-yl)-1H-indole-4-carboxamide;CS-1401;N-[(4,6-dimethyl-2-oxo-1,2-dihydro-3-pyridinyl)methyl]-3-methyl-1-[(1S)-1-methylpropyl]-6-[6-(1-piperazinyl)-3-pyridinyl]-1H-indole-4-carboxamide;GSK126||GSK-126|GSK126;GSK126;QC-9703;
分子式：C31H38N6O2
分子量：526.672
精确质量：526.306
Psa：98.8
UNII号：W4OGW9QZ97
密度：1.3±0.1g/cm3
沸点：823.4±65.0°Cat760mmHg
闪点：451.8±34.3°C
折射率：1.654
储存条件：室温，干燥，密封
蒸汽压：0.0±3.0mmHgat25°C
简介：GSK126isapotentandhighlyselectiveS-adenosyl-methionine-competitivesmallmoleculeinhibitorofEZH2methyltransferaseenzymeactivity.TheinhibitionactivityofGSK126onEZH2activitymayprovideapromisingtreatmentforEZH2mutantlymphoma.
细胞周期
