CAS号:371935-74-9
品名:N,N,N-三甲基-2-[(二甲氨基)甲酰氧基]苯铵甲磺酸盐3-(4-morpholin-4-ylpyrido[2,3]furo[2,4-b]pyrimidin-2-yl)phenol
中文别名:3-[4-(4-吗啉基吡啶并[3',2',4,5]呋喃并[3,2-D]嘧啶-2-基]苯酚盐酸盐;PI103盐酸盐;
英文别名:X6K;PI103;
分子式:C19H17ClN4O3
分子量:384.816
精确质量:384.099
Psa:84.51
MDL号:MFCD11983145
密度:1.409 g/cm3
沸点:520.25ºC at 760 mmHg
折射率:1.712
简介:PI103isadualinhbitorofClassIAphosphatidylinositol3-kinaseandmammaliantargetofrapaymycincomplex1(mTORC1),bothofwhichareinvolvedinpathwaysoftenactivatedinmyelogenousleukemia.PI103alsofunctionstoenhancetumourradiosensitivity.
PI3K/Akt/mTOR